The general formula (I) shown imidazo azines and formula (I) compound acid adduct: * * * (I) in the formula: R = 1: hydrogen, halogen, a cyano group, carboxyl, amino, nitro, formyl alkyl, halogen alkyl, alkoxy base or halogenated alkoxy, R = 2: hydrogen, halogen, nitro, cyano, carboxyl, hydroxyl, amino, mercapto, carbamoyl, sulfo, sulfamoyl chloride, or when necessary for the sulfonyl substituted alkyl, alkenyl and alkynyl, alkoxy, an oxygen radical, alkynyl oxy, alkylthio, alkene, alkyne sulfur based sulfur radical, alkyl sulfinyl, alkyl sulfonyl, amino alkyl sulfonyl, two alkyl sulfonyl amino alkyl, amino, alkyl, alkenyl two amino amino, alkynyl amino, alkyl sulfonyl amino, N - alkyl sulfonyl amino alkyl, alkoxy carbonyl, alkoxy amino sulfonyl, N alkyl alkoxy amino sulfonyl, aryl sulfonyl amino alkyl, aryl sulfonyl amide, N alkyl aryl sulfonyl amide, N alkyl aryl alkyl sulfonyl aryl sulfonyl amide, amino, aryl alkyl sulfonyl amino and N - amino alkyl aryl sulfonyl or N alkyl aryl alkyl sulfonamide group, R = 3: hydrogen, halogen, a cyano group, carboxyl, amino, hydroxyl, carbamoyl, nitro, or necessary when the substituted alkyl, alkenyl and alkynyl, alkoxy, alkene, alkyne phenoxy acetoxy, alkylthio, alkene, alkyne sulfur based sulfur radical, alkyl sulfinyl, alkyl sulfonyl, alkyl, alkenyl amide, amino alkyl alkynyl, Kiamine Based sulfonyl amino or alkoxy carbonyl, R = 4: hydrogen, halogen, alkyl, cyano or alkyl halide, R = 5: hydrogen, halogen, alkyl, cyano or alkyl halide, R = 6: halogen, cyano, nitro, amino, alkyl oxygen radicals, alkylthio, alkyl sulfinyl, alkyl sulfonyl alkyl, amino or alkyl amino two, A: C: R = n or 7 groups, D: C: R = n or 8 groups, E: C: R = n or 9 groups well, G: R = C - N or 10 groups, where R = 7, R = 8, R = 9 and R = 10. The same or different, and separate into hydrogen, halogen, a cyano group, carboxyl, carbamoyl, nitro, or necessary when all is substituted Phenyl, alkyl, alkoxy, alkylthio, alkyl sulfinyl, alkyl sulfonyl alkyl, amino, two amino alkyl or alkoxy carbonyl, with the conditions for at least one group is not up to 1 hydrogen R R = 5 group, and give up the following compounds except for: 3 - (4 - bromo 2 methyl sulfonyl phenyl) - imidazole and - 1, 2A - pyridine, 3 - bromo 2 (4 formyl phenyl) - imidazole and - 1, 2A - pyridine, 3 - bromo 2 (4 - Nitro phenyl) - imidazole and - 1. 2A - pyridine, 3 chloro 2 (4 - bromo phenyl) - imidazole and - 1, 2A - pyridine, 3 chloro 2 (4 chloro phenyl) - imidazole and - 1, 2A - pyridine, 3 Chloro 2 - (4 - methoxy phenyl) - imidazole and - 1, 2A - pyridine, 3 - bromo 2 (4 - bromo phenyl) - imidazole and - 1, 2A - pyridine, and 3 bromo 2 (4....
【技术实现步骤摘要】
本专利技术涉及新的咪唑并吖嗪类，其制备方法和其作除草剂的应用。已知，一定的2-芳基-5，6，7，8-四氢-咪唑并--吡啶具有除草的性能(参见DE-OS 41 20 108)。在文献中记载了一些咪唑并吖嗪，对其除草性能一点没公开过(参见J.Med.Chem.8(1965)，305-312—摘录于Chem.Abstracts 6216228a；Khim.Geterotsikl.Soedin 1978，258-262—摘录于Chem.Abstracts 88190733d；J.Heterocycl.Chem.25(1988)，129-137—摘录于Chem.Abstracts 11023789t；Khim.Geterotsikl.Soedin 1991，810-816—摘录于Chem.Abstracts 116128842g)。现发现一些新的通式(I)所示咪唑并吖嗪及式(I)所示化合物的酸加合物， 其中R1为氢、卤素、氰基、羧基、氨基甲酰基、硝基、烷基、卤代烷基、烷氧基或卤代烷氧基，R2为氢、卤素、氰基、羧基、硝基、羟基、巯基、氨基、氨基甲酰基、磺基、氨磺酰基、氯...
【技术保护点】
【技术特征摘要】
【专利技术属性】
技术研发人员：R·安德里，H·J·桑特尔，M·多林格，
申请(专利权)人：拜尔公司，
类型：发明
国别省市：
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